Lig221
Ligand information
- Ligand ID: Lig221
- Ligand Type : RNA
- Ligand Length : 6
- Ligand Sequence : UGGAGU
Available Structures for this Ligand- 1
| Ligand Structurename | PDB ID | Chain ID |
|---|---|---|
| 2LECB00 | 2LEC | B |
Binding Information from Structures
| Experiment ID | RRM Structure | RRM Entryename | Experiment Type | Ligand ID | Contacts |
|---|---|---|---|---|---|
| Exp_2LEC | 2LECA01 | Q01130_RRM1 | NMR | Lig221 | Contacts |
Binding Experiments for this domain - 11
| Experiment ID | RRM Entryname | Experiment Type | Ligand ID | Binds? | Binding Affinity |
|---|---|---|---|---|---|
| Exp_365 | Q01130_RRM1 | ITC | Lig221 | Yes | 0.22 ± 0.03 μM |
| Exp_367 | Q01130_RRM1 | ITC | Lig221 | Yes | 2.8 ± 0.1 μM |
| Exp_369 | Q01130_RRM1 | ITC | Lig221 | Yes | 3.7 ± 0.8 μM |
| Exp_371 | Q01130_RRM1 | ITC | Lig221 | Yes | 5 ± μM |
| Exp_373 | Q01130_RRM1 | ITC | Lig221 | Yes | 0.6 ± μM |
| Exp_376 | Q01130_RRM1 | ITC | Lig221 | No | |
| Exp_378 | Q01130_RRM1 | ITC | Lig221 | Yes | 5 ± μM |
| Exp_379 | Q01130_RRM1 | ITC | Lig221 | Yes | 0.46 ± μM |
| Exp_381 | Q01130_RRM1 | ITC | Lig221 | Yes | 0.23 ± μM |
| Exp_383 | Q01130_RRM1 | ITC | Lig221 | Yes | 0.86 ± 0.04 μM |
| Exp_385 | Q01130_RRM1 | ITC | Lig221 | Yes | 4.4 ± 0.0 μM |
RRM domains tested for Binding - 1
| RRM Entryname | Sequence Range | RRM Sequence |
|---|---|---|
| Q01130_RRM1 | 16 - 86 | LKVDNLTYRTSPDTLRRVFEKYGRVGDVYIPRDRYTKESRGFAFVRFHDKRDAEDAMDAMDGAVLDGRELR |